CP-673451

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PDGFRα/β inhibitor

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Catalog No. A11350

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
CP-673451 5mg A11350-5

Regular Price: $120.00

Special Price: $102.00

CP-673451 10mg A11350-10

Regular Price: $200.00

Special Price: $170.00

CP-673451 25mg A11350-25

Regular Price: $380.00

Special Price: $323.00

CP-673451 50mg A11350-50

Regular Price: $680.00

Special Price: $578.00

CP-673451 10mM * 1mL in DMSO A11350-10mM-D

Regular Price: $159.00

Special Price: $135.15

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

CP 673451 is a potent PDGFR-β inhibitor with an IC50 of 1 nM.

CP-673451

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Chemical Information

Catalog Num A11350
Actions Inhibitor
M. Wt 417.5
Formula C24H27N5O2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 343787-29-1
Synonyms CP673451
SMILES code COCCOC1=CC2=C(C=C1)N(C=N2)C3=NC4=C(C=CC=C4N5CCC(CC5)N)C=C3
Chemical Name 1-(2-(5-(2-methoxyethoxy)-1H-benzo[d]imidazol-1-yl)quinolin-8-yl)piperidin-4-amine

Biological Activity

Description
CP 673451 is a potent PDGFR-β inhibitor with an IC50 of 1 nM.
Targets
Target Value
PDGFRβIC50: 1nM
PDGFRαIC50: 10nM
c-KitIC50: 252nM
VEGFR1IC50: 450nM
VEGFR2IC50: 450nM
LCKIC50: >1μM
SrcIC50: >2μM
v-AblIC50: >5μM
Tie-2IC50: >5μM
bFGFRIC50: >5μM
EGFRIC50: >10μM
ErbB2IC50: >10μM
c-MetIC50: >10μM
IGF-1RIC50: >10μM

Solubility

Solubility (25°C)* In vitro DMSO 28 mg/mL heating (67.06 mM)
Water <1 mg/mL (<1 mM)
Ethanol 4 mg/mL (9.58 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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