A 922500

DGAT-1 inhibitor

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Catalog No. A11199

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
A 922500 5mg A11199-5
A 922500 10mg A11199-10
A 922500 50mg A11199-50
A 922500 100mg A11199-100
A 922500 10mM * 1mL in DMSO A11199-10mM-D

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor (IC50 values are 7 and 24 nM at human and mouse DGAT-1 respectively).

A 922500

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Chemical Information

Catalog Num A11199
Actions Inhibitor
M. Wt 428.48
Formula C26H24N2O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 959122-11-3
Synonyms DGAT-1 Inhibitor 4a, A-922500, A922500
SMILES code C1C[[email protected]]([[email protected]@H](C1)C(=O)O)C(=O)C2=CC=C(C=C2)C3=CC=C(C=C3)NC(=O)NC4=CC=CC=C4
Chemical Name (1R,2R)-2-[[4'-[[Phenylamino)carbony l]amino] [1,1'-biphenyl]-4-yl]carbonyl]cyclopentanecarboxyli c acid

Biological Activity


A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor (IC50 values are 7 and 24 nM at human and mouse DGAT-1 respectively).

human DGAT-1 mouse DGAT-1 DGAT-2
7 nM24 nM53 μM


Solubility (25°C) * In vitro DMSO 86 mg/mL (200.7 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol 20 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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