EPI-001

Androgen Receptor antagonist

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Catalog No. A15814

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
EPI-001 10mg A15814-10
$70.00
EPI-001 25mg A15814-25
$150.00
EPI-001 50mg A15814-50
$210.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 ?M)

EPI-001

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Chemical Information

Catalog Num A15814
Actions Antagonist
M. Wt 394.89
Formula C21H27ClO5
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 227947-06-0
Synonyms EPI001, EPI 001
SMILES code CC(C)(C1=CC=C(C=C1)OCC(CO)O)C2=CC=C(C=C2)OCC(CCl)O
Chemical Name 2-[4-(3-Chloro-2-hydroxypropyloxy)phenyl]-2-[4-(2,3-dihydroxypropyloxy)phenyl]propane

Biological Activity

Description
EPI-001 is an antagonist of the androgen receptor (AR) that acts by binding covalently to the N-terminal domain (NTD) of the AR and blocking protein-protein interactions required for transcriptional activity of the AR and its splice variants (IC50 for inhibition of AR NTD transactivation ?? 6 ?M)
Targets
PPARγ Androgen Receptor
N/A6 μM

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