EPZ011989

EZH2 Inhibitor

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Catalog No. A15544

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
EPZ011989 5mg A15544-5
$80.00
EPZ011989 10mg A15544-10
$140.00
EPZ011989 25mg A15544-25
$800.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.

EPZ011989

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Chemical Information

Catalog Num A15544
Actions Inhibitor
M. Wt 605.81
Formula C35H51N5O4
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 1598383-40-4
Synonyms EPZ-011989, EPZ 011989
SMILES code CCN(C1CCC(CC1)N(C)CCOC)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C#CCN4CCOCC4
Chemical Name N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl-[4-[2-methoxyethyl(methyl)amino]cyclohexyl]amino]-2-methyl-5-(3-morpholin-4-ylprop-1-ynyl)benzamide

Biological Activity

Description
EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.

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