EPZ011989

Name: EPZ011989
Brand: Adooq Bioscience
SKU: A15544
Rating: 5 (288 reviews)

Catalog No.: A15544

EZH2 Inhibitor

EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.

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Grouped product items
Size	Price	Stock
2mg	$30.00	In stock
5mg	$45.00	In stock
10mg	$70.00	In stock
25mg	$125.00	In stock
50mg	$205.00	In stock
100mg	$375.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.

Product Information

Catalog Num	A15544
Formula	C35H51N5O4
Molecular Weight	605.81
CAS Number	1598383-40-4
SMILES	CCN(C1CCC(CC1)N(C)CCOC)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C#CCN4CCOCC4
Synonyms	EPZ-011989, EPZ 011989
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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