GW842166X

CB2 receptor agonist

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Catalog No. A11253

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
GW842166X 5mg A11253-5
$60.00
GW842166X 10mg A11253-10
$100.00
GW842166X 25mg A11253-25
$200.00
GW842166X 10mM * 1mL in DMSO A11253-10mM-D
$113.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain

GW842166X

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Chemical Information

Catalog Num A11253
Actions Agonist
M. Wt 449.25
Formula C18H17Cl2F3N4O2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 666260-75-9, 956013-38-0
Synonyms N/A
SMILES code C1COCCC1CNC(=O)C2=CN=C(N=C2C(F)(F)F)NC3=C(C=C(C=C3)Cl)Cl
Chemical Name 2-(2,4-dichlorophenylamino)-N-((tetrahydro-2H-pyran-4-yl)methyl)-4-(trifluoromethyl)pyrimidine-5-carboxamide

Biological Activity

Description
GW842166X is a selective non-cannabinoid CB2 receptor agonist, which is undergoing clinical development as a novel oral treatment for inflammatory pain
Targets
CB2
63 nM(EC50)

Solubility

Solubility (25°C) * In vitro DMSO 20 mg/mL (44.51 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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