LY317615 (Enzastaurin)

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PKCβ inhibitor

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Catalog No. A10356

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
LY317615 10mg A10356-10

Regular Price: $40.00

Special Price: $32.00

LY317615 50mg A10356-50

Regular Price: $120.00

Special Price: $96.00

LY317615 100mg A10356-100

Regular Price: $200.00

Special Price: $160.00

LY317615 200mg A10356-200

Regular Price: $350.00

Special Price: $280.00

LY317615 (Enzastaurin) 10mM * 1mL in DMSO A10356-10mM-D

Regular Price: $80.00

Special Price: $64.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).

LY317615 (Enzastaurin)

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Chemical Information

Catalog Num A10356
Actions Inhibitor
M. Wt 515.6
Formula C32H29N5O2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 170364-57-5
Synonyms LY-317615
SMILES code CN1C=C(C2=CC=CC=C21)C3=C(C(=O)NC3=O)C4=CN(C5=CC=CC=C54)C6CCN(CC6)CC7=CC=CC=N7
Chemical Name 3-(1-Methylindol-3-yl)-4-[1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]indol-3-yl]pyrrole-2,5-dione

Biological Activity

Description
LY317615 (Enzastaurin) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC50= ~6 nM).
Targets
PKCβ (Cell-free assay) PKCα (Cell-free assay) PKCγ (Cell-free assay) PKCε (Cell-free assay)
6 nM39 nM83 nM110 nM

Solubility

Solubility (25°C) * In vitro DMSO 30 mg/mL (58.18 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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