PFI-2

Catalog No.: A14216
SETD7 inhibitor
PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
Grouped product items
Product Name Price Stock Qty
PFI-2 10mg
$100.00
In stock
PFI-2 25mg
$200.00
In stock
PFI-2 50mg
$350.00
In stock
PFI-2 10mM * 1mL in DMSO
$105.00
In stock
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Biological Activity
Discription PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
Targets
Target Value
Product Information
Catalog Num A14216
Formula C23H25F4N3O3S
Molecular Weight 499.52
CAS Number 1627676-59-8
SMILES C1CCN(C1)C(=O)[C@@H](CC2=CC(=CC=C2)C(F)(F)F)NS(=O)(=O)C3=CC(=C4CNCCC4=C3)F
Synonyms PFI2
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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