Rupatadine Fumarate

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PAFR inhibitor/H1 receptor inhibitor

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Catalog No. A12356

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
Rupatadine Fumarate 5mg A12356-5

Regular Price: $60.00

Special Price: $48.00

Rupatadine Fumarate 10mg A12356-10

Regular Price: $100.00

Special Price: $80.00

Rupatadine Fumarate 25mg A12356-25

Regular Price: $200.00

Special Price: $160.00

Rupatadine Fumarate 50mg A12356-50

Regular Price: $350.00

Special Price: $280.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.

Rupatadine Fumarate

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Chemical Information

Catalog Num A12356
Actions Inhibitor
M. Wt 532.03
Formula C26H26ClN3.C4H4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 182349-12-8
Synonyms N/A
SMILES code CC1=CC(=CN=C1)CN2CCC(=C3C4=C(CCC5=C3N=CC=C5)C=C(C=C4)Cl)CC2.C(=C/C(=O)O)\C(=O)O
Chemical Name 8-Chloro-6,11-dihydro-11-[1-[(5-methyl-3-pyridyl)methyl]-4-piperidylidene]-5H-benzo[5,6]cyclohepta[1,2-b]pyridine fumarate

Biological Activity

Description
Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.
Targets
Histamine H1 receptor PAFR
102 nM(Ki)550 nM(Ki)

Solubility

Solubility (25°C) * In vitro DMSO 9 mg/mL (16.91 mM)
Water <1 mg/mL (<1 mM)
Ethanol 13 mg/mL (24.43 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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