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PAFR inhibitor/H1 receptor inhibitor

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Catalog No. A11222

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
Rupatadine 5mg A11222-5

Regular Price: $80.00

Special Price: $64.00

Rupatadine 10mg A11222-10

Regular Price: $150.00

Special Price: $120.00

Rupatadine 25mg A11222-25

Regular Price: $350.00

Special Price: $280.00

Rupatadine 50mg A11222-50

Regular Price: $600.00

Special Price: $480.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.


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Chemical Information

Catalog Num A11222
Actions Inhibitor
M. Wt 415.96
Formula C26H26ClN3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 158876-82-5
Synonyms N/A
Chemical Name 8-Chloro-6,11-dihydro-11-[1-[(5-methyl-3-pyridyl)methyl]-4-piperidylidene]-5H-benzo[5,6]cyclohepta[1,2-b]pyridine

Biological Activity

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.


Solubility (25°C) * In vitro DMSO 9 mg/mL (16.91 mM)
Water <1 mg/mL (<1 mM)
Ethanol 13 mg/mL (24.43 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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