SU9516

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CDK2 inhibitor

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Catalog No. A14318

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
SU9516 10mg A14318-10

Regular Price: $90.00

Special Price: $76.50

SU9516 25mg A14318-25

Regular Price: $200.00

Special Price: $170.00

SU9516 50mg A14318-50

Regular Price: $320.00

Special Price: $272.00

SU9516 10mM * 1mL in DMSO A14318-10mM-D

Regular Price: $75.00

Special Price: $63.75

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

SU9516 is a potent, selective cdk2 inhibitor. It inhibits pRb phosphorylation causing enhanced pRB/E2F complex formation and induces G1 and G2-M cell cycle arrest.

SU9516

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Chemical Information

Catalog Num A14318
Actions Inhibitor
M. Wt 241.25
Formula C13H11N3O2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 377090-84-1
Synonyms SU 9516, SU-9516
SMILES code COC1=CC\2=C(C=C1)NC(=O)/C2=C\C3=CN=CN3
Chemical Name (Z)-1,3-Dihydro-3-(1H-imidazol-4-ylmethylene)-5-methoxy-2H-indol-2-one

Biological Activity

Description
SU9516 is a potent, selective cdk2 inhibitor. It inhibits pRb phosphorylation causing enhanced pRB/E2F complex formation and induces G1 and G2-M cell cycle arrest.
Targets
Target Value
CDK2IC50: 22nM
CDK1IC50: 40nM
CDK4IC50: 200nM
PKCIC50: >10μM
p38IC50: >10μM
PDGFRIC50: 18μM
EGFRIC50: >100μM

Solubility

Solubility (25°C)* In vitro DMSO 48 mg/mL (198.96 mM)
Water <1 mg/mL (<1 mM)
Ethanol 12 mg/mL heating (49.74 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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