UNC0379

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SETD8 HMTase inhibitor

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Catalog No. A14320

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
UNC0379 5mg A14320-5

Regular Price: $80.00

Special Price: $68.00

UNC0379 10mg A14320-10

Regular Price: $135.00

Special Price: $114.75

UNC0379 25mg A14320-25

Regular Price: $280.00

Special Price: $238.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. Its affinity to SETD8 was confirmed by ITC (isothermal titration calorimetry) and SPR (surface plasmon resonance) studies.

UNC0379

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Chemical Information

Catalog Num A14320
Actions Inhibitor
M. Wt 413.28
Formula C23H35N5O2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 1620401-82-2
Synonyms UNC-0379, UNC 0379
SMILES code COC1=C(C=C2C(=C1)C(=NC(=N2)N3CCCC3)NCCCCCN4CCCC4)OC
Chemical Name 6,7-dimethoxy-2-(pyrrolidin-1-yl)-N-(5-(pyrrolidin-1-yl)pentyl)quinazolin-4-amine

Biological Activity

Description
UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. Its affinity to SETD8 was confirmed by ITC (isothermal titration calorimetry) and SPR (surface plasmon resonance) studies.
Targets
SETD8
7.9 μM

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