APG-115

Catalog No.: A12575

MDM2 inhibitor

APG-115

APG-115 Chemical Structure

CAS NO. 1818393-16-6

APG-115 (AA-115) is an orally active MDM2 protein inhibitor binding to MDM2 protein with IC50 and Ki values of 3.8 nM and 1 nM, respectively.

Availability: In stock

Package Price Qty
1 mg

Regular Price: $320.00

Special Price $256.00

5 mg

Regular Price: $960.00

Special Price $768.00

10 mg

Regular Price: $1,600.00

Special Price $1,280.00

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Biological Activity

APG-115 (AA-115) is an orally active MDM2 protein inhibitor binding to MDM2 protein with IC50 and Ki values of 3.8 nM and 1 nM, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.56 mL 77.81 mL 155.62 mL
0.5 mM 3.11 mL 15.56 mL 31.12 mL
1 mM 1.56 mL 7.78 mL 15.56 mL
5 mM 0.31 mL 1.56 mL 3.11 mL

*The above data is based on the productmolecular weight 642.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12575
Actions Inhibitor
CAS No. 1818393-16-6
Formula C34H38Cl2FN3O4
M. Wt 642.59
Purity >98%
Synonyms APG115, APG 115
SMILES O=C1NC2=CC(Cl)=CC=C2[[email protected]]13C4(CCCCC4)N(CC)[[email protected]@H](C(NC56CCC(CC6)(C(O)=O)CC5)=O)[[email protected]@H]3C7=C(C(Cl)=CC=C7)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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