AVL-292 benzenesulfonate

Catalog No.: A15008

BTK inhibitor

AVL-292 benzenesulfonate

AVL-292 benzenesulfonate Chemical Structure

CAS NO. 1360053-81-1

AVL-292 benzenesulfonate is a covalent, highly selective, orally active small molecule inhibitor of Btk with IC50 value of 0.5 nM, >1400-fold selectivity over the other kinases assayed.

Availability: In stock

Package Price Qty
10 mg
$120.00
50 mg
$350.00
100 mg
$540.00
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Biological Activity

AVL-292 benzenesulfonate is a covalent, highly selective, orally active small molecule inhibitor of Btk with IC50 value of 0.5 nM, >1400-fold selectivity over the other kinases assayed.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.19 mL 85.97 mL 171.93 mL
0.5 mM 3.44 mL 17.19 mL 34.39 mL
1 mM 1.72 mL 8.6 mL 17.19 mL
5 mM 0.34 mL 1.72 mL 3.44 mL

*The above data is based on the productmolecular weight 581.62. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15008
Actions Inhibitor
CAS No. 1360053-81-1
Formula C28H28FN5O6S
M. Wt 581.62
Purity >98%
Synonyms AVL292 benzenesulfonate, AVL 292 benzenesulfonate
SMILES COCCOC1=CC=C(C=C1)NC2=NC=C(C(=N2)NC3=CC(=CC=C3)NC(=O)C=C)F.C1=CC=C(C=C1)S(=O)(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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