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Biological Activity
AZD-4320 is a BH3 mimetic and dual Bcl-2/Bcl-XL inhibitor.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 10.58 mL | 52.88 mL | 105.76 mL |
| 0.5 mM | 2.12 mL | 10.58 mL | 21.15 mL |
| 1 mM | 1.06 mL | 5.29 mL | 10.58 mL |
| 5 mM | 0.21 mL | 1.06 mL | 2.12 mL |
*The above data is based on the productmolecular weight 945.52. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A17171 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1357576-48-7 |
| Formula | C45H48ClF3N4O7S3 |
| M. Wt | 945.52 |
| Purity | >98% |
| Synonyms | AZD-4320, AZD-4320 |
| SMILES | O=C(NS(=O)(C1=CC=C(N[[email protected]](CCN(CCO)C)CSC2=CC=CC=C2)C(S(=O)(C(F)(F)F)=O)=C1)=O)C3=CC=C(N4CCC([[email protected]](C5=CC=CC=C5C6=CC=C(Cl)C=C6)O)CC4)C=C3 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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