BLU9931

Catalog No.: A15534

FGFR inhibitor

BLU9931

BLU9931 Chemical Structure

CAS NO. 1538604-68-0

BLU9931 is the first selective small molecule inhibitor of FGFR4 with IC50 of 3 nM; less potent for FGFR1/2/3(IC50> 150 nM),

Availability: In stock

Package Price Qty
5 mg

Regular Price: $110.00

Special Price $99.00

10 mg

Regular Price: $150.00

Special Price $135.00

25 mg

Regular Price: $220.00

Special Price $198.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

BLU9931 is the first selective small molecule inhibitor of FGFR4 with IC50 of 3 nM; less potent for FGFR1/2/3(IC50> 150 nM),
Targets
FGFR4 FGFR3 FGFR2 FGFR1
3 nM150 nM493 nM591 nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.63 mL 98.16 mL 196.32 mL
0.5 mM 3.93 mL 19.63 mL 39.26 mL
1 mM 1.96 mL 9.82 mL 19.63 mL
5 mM 0.39 mL 1.96 mL 3.93 mL

*The above data is based on the productmolecular weight 509.38. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A15534
Actions Inhibitor
M. Wt 509.38
Formula C26H22Cl2N4O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1538604-68-0
Synonyms BLU-9931, BLU 9931
SMILES CC1=C(C(=CC=C1)NC(=O)C=C)NC2=NC=C3C=C(C=CC3=N2)C4=C(C(=CC(=C4Cl)OC)OC)Cl

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