Biological Activity
FIIN-3 is a potent, selective, irreversible and the next-generation covalent FGFR inhibitor.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 14.46 mL | 72.3 mL | 144.59 mL |
0.5 mM | 2.89 mL | 14.46 mL | 28.92 mL |
1 mM | 1.45 mL | 7.23 mL | 14.46 mL |
5 mM | 0.29 mL | 1.45 mL | 2.89 mL |
*The above data is based on the productmolecular weight 691.61. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A15848 |
---|---|
Actions | Inhibitor |
CAS No. | 1637735-84-2 |
Formula | C34H36Cl2N8O4 |
M. Wt | 691.61 |
Solubility | DMSO |
Purity | >98% |
Synonyms | FIIN3, FIIN 3 |
SMILES | O=C(C=C)NC1=CC=C(CN(C2=CC(NC3=CC=C(N4CCN(C)CC4)C=C3)=NC=N2)C(NC5=C(Cl)C(OC)=CC(OC)=C5Cl)=O)C=C1 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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