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- Julia M Harrison, .et al. Muscle fiber-type specific terminal Schwann cell pathology leads to sprouting deficits following partial denervation in SOD1 G93A mice, Neurobiol Dis, 2020, Aug 20;145:105052 PMID: 32827689
Biological Activity
Masitinib mesylate is a novel inhibitor for Kit and PDGFRα/β with IC50 of 200 nM and 540 nM/800 nM, weak inhibition to ABL and c-Fms.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 16.81 mL | 84.07 mL | 168.14 mL |
| 0.5 mM | 3.36 mL | 16.81 mL | 33.63 mL |
| 1 mM | 1.68 mL | 8.41 mL | 16.81 mL |
| 5 mM | 0.34 mL | 1.68 mL | 3.36 mL |
*The above data is based on the productmolecular weight 594.75. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A15152 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1048007-93-7 |
| Formula | C29H34N6O4S2 |
| M. Wt | 594.75 |
| Purity | >98% |
| Synonyms | AB1010 mesylate, Masivet mesylate, AB-1010 mesylate, AB 1010 mesylate |
| SMILES | CC1=C(C=C(C=C1)NC(=O)C2=CC=C(C=C2)CN3CCN(CC3)C)NC4=NC(=CS4)C5=CN=CC=C5.CS(=O)(=O)O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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