Masitinib mesylate

Catalog No.: A15152

KIT/PDGFR inhibitor

Masitinib mesylate

Masitinib mesylate Chemical Structure

CAS NO. 1048007-93-7

Masitinib mesylate is a novel inhibitor for Kit and PDGFRα/β with IC50 of 200 nM and 540 nM/800 nM, weak inhibition to ABL and c-Fms.

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50 mg
$100.00
200 mg
$250.00
500 mg
$470.00
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  • Julia M Harrison, .et al. Muscle fiber-type specific terminal Schwann cell pathology leads to sprouting deficits following partial denervation in SOD1 G93A mice, Neurobiol Dis, 2020, Aug 20;145:105052 PMID: 32827689

Biological Activity

Masitinib mesylate is a novel inhibitor for Kit and PDGFRα/β with IC50 of 200 nM and 540 nM/800 nM, weak inhibition to ABL and c-Fms.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.81 mL 84.07 mL 168.14 mL
0.5 mM 3.36 mL 16.81 mL 33.63 mL
1 mM 1.68 mL 8.41 mL 16.81 mL
5 mM 0.34 mL 1.68 mL 3.36 mL

*The above data is based on the productmolecular weight 594.75. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15152
Actions Inhibitor
CAS No. 1048007-93-7
Formula C29H34N6O4S2
M. Wt 594.75
Purity >98%
Synonyms AB1010 mesylate, Masivet mesylate, AB-1010 mesylate, AB 1010 mesylate
SMILES CC1=C(C=C(C=C1)NC(=O)C2=CC=C(C=C2)CN3CCN(CC3)C)NC4=NC(=CS4)C5=CN=CC=C5.CS(=O)(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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