PF-04217903 phenolsulfonate

Catalog No.: A34328
c-Met inhibitor
PF-04217903 phenolsulfonate is a potent ATP-competitive inhibitor of the c-Met kinase with a Ki value of 4.8 nM for human c-Met. It demonstrates over 1,000-fold selectivity against a profile of 208 kinases, highlighting its specificity. This compound possesses antiangiogenic properties and is useful in research applications related to cancer therapy and the modulation of tumor microenvironments.
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Adooq Products cited in reputable paper
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Biological Activity
DescriptionPF-04217903 phenolsulfonate is a potent ATP-competitive inhibitor of the c-Met kinase with a Ki value of 4.8 nM for human c-Met. It demonstrates over 1,000-fold selectivity against a profile of 208 kinases, highlighting its specificity. This compound possesses antiangiogenic properties and is useful in research applications related to cancer therapy and the modulation of tumor microenvironments.
Product Information
Catalog NumA34328
FormulaC25H22N8O5S
Molecular Weight546.56
CAS Number1159490-85-3
SMILESO=S(C1=CC=C(O)C=C1)(O)=O.OCCN2N=CC(C3=CN=C4C(N(CC5=CC=C6N=CC=CC6=C5)N=N4)=N3)=C2
Useful Calculator

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Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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