TAK 259

Catalog No.: A16186

α1D Adrenoceptor Antagonist

TAK 259

TAK 259 Chemical Structure

CAS NO. 1192347-42-4

TAK-259 is a Novel, Selective, and Orally Active α1D Adrenoceptor Antagonist (α1D, Ki = 1.1 nM) with Anti-urinary Frequency Effects and Reducing Human Ether-a-go-go-Related Gene (hERG) Liabilities.

Availability: In stock

Package Price Qty
10 mg
$90.00
25 mg
$180.00
100 mg
$540.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

TAK-259 is a Novel, Selective, and Orally Active α1D Adrenoceptor Antagonist (α1D, Ki = 1.1 nM) with Anti-urinary Frequency Effects and Reducing Human Ether-a-go-go-Related Gene (hERG) Liabilities.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.35 mL 121.74 mL 243.49 mL
0.5 mM 4.87 mL 24.35 mL 48.7 mL
1 mM 2.43 mL 12.17 mL 24.35 mL
5 mM 0.49 mL 2.43 mL 4.87 mL

*The above data is based on the productmolecular weight 410.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A16186
Actions Antagonist
M. Wt 410.7
Formula C14H14Cl3N3O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1192347-42-4
Synonyms TAK259, TAK-259
SMILES O=C(C1=CC(Cl)=CN(CC2=CC(Cl)=CC=C2S(=O)(C)=O)C1=N)N.[H]Cl

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