WH 4-023

Catalog No.: A14117

dual Lck/Src inhibitor

WH 4-023 Chemical Structure

CAS NO. 837422-57-8

WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC50 of 2 nM/6 nM for Lck and Src kinase respectively.

Availability: In stock

Package Price Qty
10 mg
$120.00
25 mg
$250.00
50 mg
$400.00
10mM * 1mL in DMSO
$100.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC50 of 2 nM/6 nM for Lck and Src kinase respectively.
Targets
Lck (Cell-free assay) Src (Cell-free assay)
2 nM6 nM
In vitro DMSO 12 mg/mL heating (21.1 mM)
Water <1 mg/mL (<1 mM)
Ethanol 6 mg/mL heating (10.55 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.58 mL 87.92 mL 175.85 mL
0.5 mM 3.52 mL 17.58 mL 35.17 mL
1 mM 1.76 mL 8.79 mL 17.58 mL
5 mM 0.35 mL 1.76 mL 3.52 mL

*The above data is based on the productmolecular weight 568.67. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14117
Actions Inhibitor
M. Wt 568.67
Formula C32H36N6O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 837422-57-8
Synonyms WH-4-023,WH4-023
SMILES CC1=C(C(=CC=C1)C)OC(=O)N(C2=C(C=C(C=C2)OC)OC)C3=NC(=NC=C3)NC4=CC=C(C=C4)N5CCN(CC5)C

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