AS-605240

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PI3K Inhibitor

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Catalog No. A10088

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
AS-605240 10mg A10088-10

Regular Price: $40.00

Special Price: $32.00

AS-605240 25mg A10088-25

Regular Price: $100.00

Special Price: $80.00

AS-605240 50mg A10088-50

Regular Price: $180.00

Special Price: $144.00

AS-605240 100mg A10088-100

Regular Price: $260.00

Special Price: $208.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

AS-605240 is an orally active inhibitor of PI3-kinase γ that inhibits human recombinant PI3Kγ, α, β, and δ in an ATP-competitive manner with IC50 values of 8, 60, 270, and 300 nM, respectively.

AS-605240

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Chemical Information

Catalog Num A10088
Actions Inhibitor
M. Wt 257.3
Formula C12H7N3O2S
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 648450-29-7
Synonyms AS605240
SMILES code C1=CC2=NC=CN=C2C=C1/C=C\3/C(=O)NC(=O)S3
Chemical Name 5-(6-Quinoxalinylmethylene)-2,4-thiazolidine-2,4-dione

Biological Activity

Description
AS-605240 is an orally active inhibitor of PI3-kinase γ that inhibits human recombinant PI3Kγ, α, β, and δ in an ATP-competitive manner with IC50 values of 8, 60, 270, and 300 nM, respectively.
Targets
PI3Kγ (Cell-free assay) PI3Kα (Cell-free assay) PI3Kβ (Cell-free assay) PI3Kδ (Cell-free assay)
8 nM60 nM270 nM300 nM

Solubility

Solubility (25°C) * In vitro DMSO 0.4 mg/mL (1.55 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 0.5% CMC/0.25% Tween 80 11 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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