CH5132799

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PI3K inhibitor

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Catalog No. A11169

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
CH5132799 5mg A11169-5

Regular Price: $180.00

Special Price: $144.00

CH5132799 10mg A11169-10

Regular Price: $280.00

Special Price: $224.00

CH5132799 50mg A11169-50

Regular Price: $780.00

Special Price: $624.00

CH5132799 100mg A11169-100

Regular Price: $1,100.00

Special Price: $880.00

CH5132799 10mM * 1mL in DMSO A11169-10mM-D

Regular Price: $195.00

Special Price: $156.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

CH5132799 is a novel class I PI3K inhibitor, which exhibited a strong inhibitory activity especially against PI3Kα (IC(50)=0.014 μM).

CH5132799

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Chemical Information

Catalog Num A11169
Actions Inhibitor
M. Wt 377.42
Formula C15H19N7O3S
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 1007207-67-1
Synonyms CH-5132799
SMILES code CS(=O)(=O)N1CCC2=C(N=C(N=C21)N3CCOCC3)C4=CN=C(N=C4)N
Chemical Name 5-(7-(methylsulfonyl)-2-morpholino-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrimidin-2-amine

Biological Activity

Description

CH5132799 is a novel class I PI3K inhibitor, which exhibited a strong inhibitory activity especially against PI3Kα (IC(50)=0.014 μM).

Targets
Target Value
PI3KαIC50: 14nM
PI3KγIC50: 36nM
PI3KβIC50: 0.12μM
PI3KδIC50: 0.50μM
mTORIC50: 1.6μM
C2βIC50: 5.3μM
C2αIC50: >10μM
Vps34IC50: >10μM

Solubility

Solubility (25°C) * In vitro DMSO 12 mg/mL (31.79 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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