G007-LK

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TNKS inhibitor

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Catalog No. A15528

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
G007-LK 5mg A15528-5

Regular Price: $80.00

Special Price: $68.00

G007-LK 10mg A15528-10

Regular Price: $140.00

Special Price: $119.00

G007-LK 25mg A15528-25

Regular Price: $300.00

Special Price: $255.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

G007-LK displays high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice,

G007-LK

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Chemical Information

Catalog Num A15528
Actions Inhibitor
M. Wt 529.96
Formula C25H16ClN7O3S
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 1380672-07-0
Synonyms G007 LK, G007LK
SMILES code CS(=O)(=O)C1=CN=C(C=C1)C2=NN=C(N2C3=CC=CC=C3Cl)C=CC4=NN=C(O4)C5=CC=C(C=C5)C#N
Chemical Name (E)-4-(5-(2-(4-(2-chlorophenyl)-5-(5-(methylsulfonyl)pyridin-2-yl)-4H-1,2,4-triazol-3-yl)vinyl)-1,3,4-oxadiazol-2-yl)benzonitrile

Biological Activity

Description
G007-LK displays high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice,
Targets

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