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GSK 525762A (I-BET-762)


BET inhibitor

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Catalog No. A11440

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
GSK 525762A 5mg A11440-5

Regular Price: $80.00

Special Price: $72.00

GSK 525762A 10mg A11440-10

Regular Price: $120.00

Special Price: $108.00

GSK 525762A 25mg A11440-25

Regular Price: $240.00

Special Price: $216.00

GSK 525762A 50mg A11440-50

Regular Price: $360.00

Special Price: $324.00

GSK 525762A (I-BET-762) 10mM * 1mL in DMSO A11440-10mM-D

Regular Price: $90.00

Special Price: $81.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

GSK-525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family

GSK 525762A (I-BET-762)

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Chemical Information

Catalog Num A11440
Actions Inhibitor
M. Wt 423.9
Formula C22H22ClN5O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1260907-17-2
Synonyms GSK-525762A, GSK525762A
SMILES code CCNC(=O)C[[email protected]]1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C
Chemical Name (4S)-6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide

Biological Activity

GSK-525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family
BET proteins (Cell-free assay)
35 nM


Solubility (25°C)* In vitro DMSO 84 mg/mL (198.15 mM)
Water <1 mg/mL (<1 mM)
Ethanol 84 mg/mL (198.15 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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