Molibresib besylate

Catalog No.: A21855

BET bromodomain inhibitor

Molibresib besylate

Molibresib besylate Chemical Structure

CAS NO. 1895049-20-3

Molibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM.

Availability: In stock

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5 mg

Regular Price: $95.00

Special Price $76.00

10 mg

Regular Price: $164.00

Special Price $131.20

50 mg

Regular Price: $488.00

Special Price $390.40

100 mg

Regular Price: $975.00

Special Price $780.00

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Biological Activity

Molibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.18 mL 85.9 mL 171.8 mL
0.5 mM 3.44 mL 17.18 mL 34.36 mL
1 mM 1.72 mL 8.59 mL 17.18 mL
5 mM 0.34 mL 1.72 mL 3.44 mL

*The above data is based on the productmolecular weight 582.07. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21855
Actions Inhibitor
CAS No. 1895049-20-3
Formula C28H28ClN5O5S
M. Wt 582.07
Purity >98%
Synonyms GSK 525762C, GSK-525762C, GSK525762C; I-BET 762 besylate, I-BET762, I-BET-762
SMILES ClC1=CC=C(C2=N[[email protected]@H](CC(NCC)=O)C3=NN=C(C)N3C4=CC=C(OC)C=C24)C=C1.O=S(C5=CC=CC=C5)(O)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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