Kenpaullone

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CDK inhibitor

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Catalog No. A11220

Availability:Stock in USAIn stock Shipped in 7-10 Days

Product Name Catalog No. Price Qty
Kenpaullone 10mg A11220-10

Regular Price: $90.00

Special Price: $72.00

Kenpaullone 50mg A11220-50

Regular Price: $380.00

Special Price: $304.00

Kenpaullone 100mg A11220-100

Regular Price: $650.00

Special Price: $520.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases.

Kenpaullone

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Chemical Information

Catalog Num A11220
Actions Inhibitor
M. Wt 327.2
Formula C16H11BrN2O
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 142273-20-9
Synonyms N/A
SMILES code C1C2=C(C3=CC=CC=C3NC1=O)NC4=C2C=C(C=C4)Br
Chemical Name 9-Bromo-7,12-dihydro-indolo[3,2-d][1]benzazepin-6(5H)-one

Biological Activity

Description
Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases.
Targets
Target Value
GSK-3βIC50: 0.23μM
CDK1/CyclinBIC50: 0.4μM
CDK2/CyclinAIC50: 0.68μM
CDK5/p35IC50: 0.85μM
CDK2/CyclinEIC50: 7.5μM
ERK2IC50: 9μM
c-SrcIC50: 15μM
CaseinKinase2IC50: 20μM
ERK1IC50: 20μM

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