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LB42708

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FTase inhibitor

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Catalog No. A14020

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
LB42708 5mg A14020-5

Regular Price: $60.00

Special Price: $48.00

LB42708 10mg A14020-10

Regular Price: $100.00

Special Price: $80.00

LB42708 25mg A14020-25

Regular Price: $200.00

Special Price: $160.00

LB42708 10mM * 1mL in DMSO A14020-10mM-D

Regular Price: $126.00

Special Price: $100.80

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

LB42708 is a potent, orally active and selective nonpeptidic farnesyltransferase inhibitor (FTase inhibitor).

LB42708

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Chemical Information

Catalog Num A14020
Actions Inhibitor
M. Wt 555.46
Formula C30H27BrN4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 226929-39-1
Synonyms LB-42708, LB 42708
SMILES code C1COCCN1C(=O)C2=CN(C=C2C3=CC=CC4=CC=CC=C43)CC5=CN=CN5CC6=CC=C(C=C6)Br
Chemical Name (1-((1-(4-bromobenzyl)-1H-imidazol-5-yl)methyl)-4-(naphthalen-1-yl)-1H-pyrrol-3-yl)(morpholino)methanone

Biological Activity

Description
LB42708 is a potent, orally active and selective nonpeptidic farnesyltransferase inhibitor (FTase inhibitor).
Targets
FTase (H-ras) FTase (N-ras) FTase (K-Ras)
0.8 nM1.2 nM2.0 nM

Solubility

Solubility (25°C)* In vitro DMSO 100 mg/mL (180.03 mM)
Water <1 mg/mL (<1 mM)
Ethanol 86 mg/mL heating (154.82 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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