P005091

DUB/USP7 Inhibitor

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Catalog No. A13277

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
P005091 10mg A13277-10

Regular Price: $80.00

Special Price: $68.00

P005091 25mg A13277-25

Regular Price: $170.00

Special Price: $144.50

P005091 50mg A13277-50

Regular Price: $250.00

Special Price: $212.50

P005091 10mM * 1mL in DMSO A13277-10mM-D

Regular Price: $89.00

Special Price: $75.65

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

P005091 is a selective inhibitor of ubiquitin-specific protease (USP) 7 (IC50 = 4.2 uM).

P005091

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Chemical Information

Catalog Num A13277
Actions Inhibitor
M. Wt 348.22
Formula C12H7Cl2NO3S2
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 882257-11-6
Synonyms P5091
SMILES code CC(=O)C1=CC(=C(S1)SC2=C(C(=CC=C2)Cl)Cl)[N+](=O)[O-]
Chemical Name 1-[5-[(2,3-Dichlorophenyl)thio]-4-nitro-2-thienyl]ethanone

Biological Activity

Description
P005091 is a selective inhibitor of ubiquitin-specific protease (USP) 7 (IC50 = 4.2 uM).
Targets
Target Value
USP7EC504.2μM
Calpain1EC50>100μM
MMP13EC50>100μM
CathepsinDEC50>100μM
EKLEC50>100μM
PLA2EC50>100μM
USP2cEC50>100μM
USP5EC50>100μM
USP8cEC50>100μM
USP15EC50>100μM
USP20EC50>100μM
USP21EC50>100μM
USP28EC50>100μM
UCH-L1EC50>100μM
Caspase-3EC50>100μM
CathepsinKEC50>100μM

Solubility

Solubility (25°C) * In vitro DMSO 28 mg/mL (80.4 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol, pH 4 10 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

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