Biological Activity
Mps1-IN-1 is a highly potent and selectibe Mpsl inhibitor with IC50 of 367 nM; >1000-fold selectivity relative to the 352 member kinase panel with the major exceptions of Alk and Ltk.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 18.67 mL | 93.34 mL | 186.69 mL |
0.5 mM | 3.73 mL | 18.67 mL | 37.34 mL |
1 mM | 1.87 mL | 9.33 mL | 18.67 mL |
5 mM | 0.37 mL | 1.87 mL | 3.73 mL |
*The above data is based on the productmolecular weight 535.66. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A11218 |
---|---|
Actions | Inhibitor |
CAS No. | 1125593-20-5 |
Formula | C28H33N5O4S |
M. Wt | 535.66 |
Purity | >98% |
SMILES | OC1CCN(C2=CC(OC)=C(NC3=NC4=C(C=CN4)C(NC5=C(S(=O)(C(C)C)=O)C=CC=C5)=C3)C=C2)CC1 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy Mps1-IN-1 | Mps1-IN-1 Supplier | purchase | cost | manufacturer | order | distributor | buy 1125593-20-5| 1125593-20-5 Supplier | purchase 1125593-20-5 | 1125593-20-5 cost | 1125593-20-5 manufacturer | order 1125593-20-5 | 1125593-20-5 distributor