Fig. 1 · Structure
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2,6-Dimethylquinoline
Cat. No.
A69741
CAS
877-43-0
CYP1A2 Inhibitor
2,6-Dimethylquinoline is a selective inhibitor of CYP1A2, exhibiting an IC50 of 3.3 µM. Additionally, it shows inhibitory activity towards CYP2B6 with an IC50 of 480 µM. This compound, derived from the roots of Peucedanum praeruptorum, serves as a valuable tool for research into drug metabolism and pharmacokinetics, particularly in studies exploring cytochrome P450 enzyme modulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 877-43-0 |
| Applications | CYP1A2 Inhibitor |
| Formula | C11H11N |
| Molecular Weight | 157.22 |
| SMILES | CC1=CC2=C(C=C1)N=C(C)C=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.