A 803467

Catalog No.: A11234

Sodium channel Blocker

A 803467

A 803467 Chemical Structure

CAS NO. 944261-79-4

A 803467 is a selective blocker of NaV1.8 channels (IC50 values are 8, 2450, 6740, 7340 and 7380 nM for hNaV1.8, hNaV1.3, hNaV1.7, hNaV1.5 and hNaV1.2 channels respectively).

Availability: In stock

Package Price Qty
10 mg

Regular Price: $50.00

Special Price $40.00

25 mg

Regular Price: $98.00

Special Price $78.40

50 mg

Regular Price: $150.00

Special Price $120.00

100 mg

Regular Price: $250.00

Special Price $200.00

10mM * 1mL in DMSO
$77.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

A 803467 is a selective blocker of NaV1.8 channels (IC50 values are 8, 2450, 6740, 7340 and 7380 nM for hNaV1.8, hNaV1.3, hNaV1.7, hNaV1.5 and hNaV1.2 channels respectively).
Targets
Na(V1.8) channel
8 nM
In vitro (25°C) DMSO 72 mg/mL (201.23 mM)
Water <1 mg/mL (<1 mM)
Ethanol 11 mg/mL (30.74 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.95 mL 139.74 mL 279.49 mL
0.5 mM 5.59 mL 27.95 mL 55.9 mL
1 mM 2.79 mL 13.97 mL 27.95 mL
5 mM 0.56 mL 2.79 mL 5.59 mL

*The above data is based on the productmolecular weight 357.8. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A11234
Actions Blocker
M. Wt 357.8
Formula C19H16ClNO4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 944261-79-4
Synonyms A-803467, A803467
SMILES COC1=CC(=CC(=C1)NC(=O)C2=CC=C(O2)C3=CC=C(C=C3)Cl)OC

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