A1/A3 AR antagonist 3

Catalog No.: A57952
A1R/A3R Dual Antagonist
A1/A3 AR Antagonist 3 is a dual antagonist targeting A1 and A3 adenosine receptors, exhibiting high affinity in the low-micromolar to low-nanomolar range. This compound is instrumental in researching chronic heart diseases, facilitating the exploration of mechanisms involved in cardiac function and pathology. Its selective inhibition of A1 and A3 receptors may provide insights into potential therapeutic strategies for related cardiovascular disorders.
Grouped product items
Size Price Stock Qty
25mg
$1,530.00
In stock
50mg
$1,950.00
In stock
100mg
$2,480.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

Loading distributor info...

Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionA1/A3 AR Antagonist 3 is a dual antagonist targeting A1 and A3 adenosine receptors, exhibiting high affinity in the low-micromolar to low-nanomolar range. This compound is instrumental in researching chronic heart diseases, facilitating the exploration of mechanisms involved in cardiac function and pathology. Its selective inhibition of A1 and A3 receptors may provide insights into potential therapeutic strategies for related cardiovascular disorders.
Product Information
Catalog NumA57952
FormulaC22H19N5O3
Molecular Weight401.42
CAS Number2665804-57-7
SMILESN#CC1=CC2=C(NN=C2C3=CC=CC=C3)C(NC4=CC(OC)=C(C(OC)=C4)OC)=N1
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2