A2A receptor antagonist 1

Catalog No.: A12567

adenosine A2A/A1 receptor antagonist

A2A receptor antagonist 1

A2A receptor antagonist 1 Chemical Structure

CAS NO. 443103-97-7

A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.

Availability: In stock

Package Price Qty
1 mg
$45.00
5 mg
$135.00
10 mg
$230.00
50 mg
$690.00
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Biological Activity

A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
In vitro DMSO 60 mg/mL (193.98 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 32.33 mL 161.66 mL 323.31 mL
0.5 mM 6.47 mL 32.33 mL 64.66 mL
1 mM 3.23 mL 16.17 mL 32.33 mL
5 mM 0.65 mL 3.23 mL 6.47 mL

*The above data is based on the productmolecular weight 309.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12567
Actions Antagonist
CAS No. 443103-97-7
Formula C16H12FN5O
M. Wt 309.3
Purity >98%
Synonyms CPI-444 analog, CPI444, CPI 444
SMILES NC1=NC(C2=CC=CO2)=C3C(N(CC4=C(F)C=CC=C4)N=C3)=N1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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