Acolbifene (EM 652, SCH57068)

Catalog No.: A12771

estrogen receptor modulator

Acolbifene (EM 652, SCH57068)

Acolbifene (EM 652, SCH57068) Chemical Structure

CAS NO. 182167-02-8

acolbifene is a substance being studied in the prevention of breast cancer in women at high risk of breast cancer. Acolbifene hydrochloride binds to estrogen receptors in the body and blocks the effects of estrogen in the breast. It is a type of selective estrogen receptor modulator (SERM).

Availability: In stock

Package Price Qty
5 mg

Regular Price: $350.00

Special Price $280.00

10 mg

Regular Price: $650.00

Special Price $520.00

25 mg

Regular Price: $1,200.00

Special Price $960.00

50 mg

Regular Price: $2,000.00

Special Price $1,600.00

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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Sumit Bansal, .et al. Inhibition of Human Sulfotransferase 2A1-Catalyzed Sulfonation of Lithocholic Acid, Glycolithocholic Acid, and Taurolithocholic Acid by Selective Estrogen Receptor Modulators and Various Analogs and Metabolites, J Pharmacol Exp Ther, 2019, June, 369 (3) 389-405
  • Lirit N. Franks, .et al. Selective Estrogen Receptor Modulators: Cannabinoid Receptor Inverse Agonists with Differential CB1 and CB2 Selectivity, Front Pharmacol, 2016, 7: 503 PMID: 28066250

Biological Activity

acolbifene is a substance being studied in the prevention of breast cancer in women at high risk of breast cancer. Acolbifene hydrochloride binds to estrogen receptors in the body and blocks the effects of estrogen in the breast. It is a type of selective estrogen receptor modulator (SERM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.86 mL 109.28 mL 218.55 mL
0.5 mM 4.37 mL 21.86 mL 43.71 mL
1 mM 2.19 mL 10.93 mL 21.86 mL
5 mM 0.44 mL 2.19 mL 4.37 mL

*The above data is based on the productmolecular weight 457.56. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12771
Actions Modulator
CAS No. 182167-02-8
Formula C29H31NO4
M. Wt 457.56
Purity >98%
Synonyms EM652, EM-652, SCH-57068, SCH 57068
SMILES CC1=C([[email protected]@H](OC2=C1C=CC(=C2)O)C3=CC=C(C=C3)OCCN4CCCCC4)C5=CC=C(C=C5)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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