Adenosine receptor inhibitor 2

Catalog No.: A57913
AR Inhibitor
Adenosine receptor inhibitor 2 (compound 14b) is a selective antagonist of adenosine receptors, primarily targeting A1 and A2A subtypes. This compound exhibits a higher affinity for A1AR, with a Ki value of 52.2 nM, compared to 167 nM for A2AAR. Its potent inhibitory effects make it valuable for research exploring adenosine signaling pathways, and its applications may extend to studies in cardiovascular disease, cancer, and neurobiology.
Grouped product items
Size Price Stock Qty
1mg
$360.00
In stock
5mg
$825.00
In stock
10mg
$1,010.00
In stock
25mg
$1,275.00
In stock
50mg
$1,625.00
In stock
100mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionAdenosine receptor inhibitor 2 (compound 14b) is a selective antagonist of adenosine receptors, primarily targeting A1 and A2A subtypes. This compound exhibits a higher affinity for A1AR, with a Ki value of 52.2 nM, compared to 167 nM for A2AAR. Its potent inhibitory effects make it valuable for research exploring adenosine signaling pathways, and its applications may extend to studies in cardiovascular disease, cancer, and neurobiology.
Product Information
Catalog NumA57913
FormulaC17H20BrN5O2
Molecular Weight406.28
CAS Number2550401-76-6
SMILESO=C(N1CC)N(CC)C2=C(N(C)C(NCC3=CC=CC(Br)=C3)=N2)C1=O
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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