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Ala1,3,11,15-Endothelin (53-63)

Catalog No.: A60256
ETB Agonist
[Ala1,3,11,15]-Endothelin (53-63) is a selective agonist for the ETB receptor, exhibiting potent activity with IC50 values between 0.33 nM and 0.61 nM. This compound is valuable for research focused on vasoconstriction and related physiological processes. Its specificity for the ETB receptor makes it a useful tool for investigating the role of endothelins in vascular biology and potential therapeutic applications.
[Ala1,3,11,15]-Endothelin (53-63) 121204-87-3 ETB Agonist
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Size Price Stock Qty
5mg
$410.00
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
Description[Ala1,3,11,15]-Endothelin (53-63) is a selective agonist for the ETB receptor, exhibiting potent activity with IC50 values between 0.33 nM and 0.61 nM. This compound is valuable for research focused on vasoconstriction and related physiological processes. Its specificity for the ETB receptor makes it a useful tool for investigating the role of endothelins in vascular biology and potential therapeutic applications.
Product Information
Catalog NumA60256
FormulaC109H163N25O32S
Molecular Weight2367.67
CAS Number121204-87-3
Sequence shorteningASASSLMDKEAVYFAHLDIIW
SMILESC([C@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC1=CN=CN1)NC([C@@H](NC([C@H](CC2=CC=CC=C2)NC([C@H](CC3=CC=C(O)C=C3)NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](C)N)=O)CO)=O)C)=O)CO)=O)CO)=O)CC(C)C)=O)CCSC)=O)CC(O)=O)=O)CCCCN)=O)CCC(O)=O)=O)C)=O)C(C)C)=O)=O)=O)C)=O)=O)CC(C)C)=O)CC(O)=O)=O)[C@H](CC)C)=O)[C@H](CC)C)=O)C(O)=O)C=4C=5C(NC4)=CC=CC5
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GPCR/G Protein > Endothelin Receptors