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Ambrisentan (BSF 208075)


EndothelinA receptor antagonist

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Catalog No. A11291

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
Ambrisentan 5mg A11291-5

Regular Price: $50.00

Special Price: $45.00

Ambrisentan 10mg A11291-10

Regular Price: $60.00

Special Price: $54.00

Ambrisentan 25mg A11291-25

Regular Price: $110.00

Special Price: $99.00

Ambrisentan 50mg A11291-50

Regular Price: $190.00

Special Price: $171.00

Ambrisentan (BSF 208075) 10mM * 1mL in DMSO A11291-10mM-D

Regular Price: $50.00

Special Price: $45.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Ambrisentan functions as an endothelin receptor antagonist, and is selective for the type A endothelin receptor (ETA).

Ambrisentan (BSF 208075)

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Publications citing Adooq Products
Ambrisentan (BSF 208075) Citations (2)
  • Tony Ngo, .et al. Orphan receptor ligand discovery by pickpocketing pharmacological neighbors, Nat Chem Biol, 2017, Feb; 13(2): 235-242 PMID: 27992882
  • Toshiaki Okamoto, .et al. Antifibrotic effects of ambrisentan, an endothelin-A receptor antagonist, in a non-alcoholic steatohepatitis mouse model, World J Hepatol, 2016, Aug 8; 8(22): 933-941 PMID: 27574547

Chemical Information

Catalog Num A11291
Actions Antagonist
M. Wt 378.4
Formula C22H22N2O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 177036-94-1
Synonyms BSF 208075,
SMILES CC1=CC(=NC(=N1)O[[email protected]](C(=O)O)C(C2=CC=CC=C2)(C3=CC=CC=C3)OC)C

Biological Activity

Ambrisentan functions as an endothelin receptor antagonist, and is selective for the type A endothelin receptor (ETA).


Solubility (25°C)* In vitro DMSO 76 mg/mL (200.83 mM)
Water <1 mg/mL (<1 mM)
Ethanol 22 mg/mL (58.13 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.43 mL 132.14 mL 264.27mL
0.5 mM 5.29 mL 26.43 mL 52.85 mL
1 mM 2.64 mL 13.21 mL 26.43 mL
5 mM 0.53 mL 2.64 mL 5.29 mL

*The above data is based on the productmolecular weight 378.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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