Antihistamine-1

Name: Antihistamine-1
Brand: Adooq Bioscience
SKU: A20515
Rating: 5 (288 reviews)

Catalog No.: A20515

Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.

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Grouped product items
Size	Price	Stock
1mg	$20.00	In stock
5mg	$45.00	In stock
10mg	$85.00	In stock
25mg	$180.00	In stock
50mg	$345.00	In stock
100mg	$650.00	In stock
*10mM 1mL in DMSO**	$50.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description

Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

Product Information

Catalog Num	A20515
Formula	C23H24FN5
Molecular Weight	389.47
CAS Number	1186430-60-3
SMILES	CC1=CN(C2CCN(C3=NC4=CC=CC=C4N3CC5=CC=C(F)C=C5)CC2)N=C1
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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