AP-238

Catalog No.: A62502
MOR Agonist
AP-238 is a synthetic opioid that primarily targets the μ-opioid receptor (MOR), exhibiting an EC50 value of 248 nM. This compound demonstrates significant analgesic properties, making it relevant for research focused on pain management and opioid receptor pharmacology. Its ability to activate MOR positions AP-238 as a valuable tool for studying the effects of opioids in various biological contexts.
Grouped product items
Size Price Stock Qty
5mg
$350.00
In stock
10mg
$650.00
In stock
50mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionAP-238 is a synthetic opioid that primarily targets the μ-opioid receptor (MOR), exhibiting an EC50 value of 248 nM. This compound demonstrates significant analgesic properties, making it relevant for research focused on pain management and opioid receptor pharmacology. Its ability to activate MOR positions AP-238 as a valuable tool for studying the effects of opioids in various biological contexts.
Product Information
Catalog NumA62502
FormulaC18H26N2O
Molecular Weight286.41
CAS Number140924-11-4
SMILESCCC(N1[C@H](C)CN(C/C=C/C2=CC=CC=C2)C[C@@H]1C)=O
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