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APS-2-79 HCl, small molecule that stabilizes the KSR (Kinase suppressor of Ras) inactive state and antagonizes oncogenic Ras signalling (IC50 value 120 nM against ATP-biotin probe-labelling of KSR2).
Targets
| KSR2 | ||||
| 120 nM |
| In vitro | DMSO | 82 mg/mL (193.44 mM) | |
| Water | Insoluble | ||
| Ethanol | 27 mg/mL (63.69 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.59 mL | 117.96 mL | 235.91 mL |
| 0.5 mM | 4.72 mL | 23.59 mL | 47.18 mL |
| 1 mM | 2.36 mL | 11.8 mL | 23.59 mL |
| 5 mM | 0.47 mL | 2.36 mL | 4.72 mL |
*The above data is based on the productmolecular weight 423.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A16175 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 2002381-31-7 |
| Formula | C23H21N3O3.HCl |
| M. Wt | 423.89 |
| Purity | >98% |
| Synonyms | KSR/Ras Inhibitor |
| SMILES | CC1=C(C=CC(=C1)OC2=CC=CC=C2)NC3=NC=NC4=CC(=C(C=C43)OC)OC.Cl |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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