APS-2-79 HCl

Catalog No.: A16175

KSR/Ras inhibitor

APS-2-79 HCl

APS-2-79 HCl Chemical Structure

CAS NO. 2002381-31-7

APS-2-79 HCl, small molecule that stabilizes the KSR (Kinase suppressor of Ras) inactive state and antagonizes oncogenic Ras signalling (IC50 value 120 nM against ATP-biotin probe-labelling of KSR2).

Availability: In stock

Package Price Qty
5 mg
$90.00
10 mg
$160.00
50 mg
$620.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

APS-2-79 HCl, small molecule that stabilizes the KSR (Kinase suppressor of Ras) inactive state and antagonizes oncogenic Ras signalling (IC50 value 120 nM against ATP-biotin probe-labelling of KSR2).
Targets
KSR2
120 nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.59 mL 117.96 mL 235.91 mL
0.5 mM 4.72 mL 23.59 mL 47.18 mL
1 mM 2.36 mL 11.8 mL 23.59 mL
5 mM 0.47 mL 2.36 mL 4.72 mL

*The above data is based on the productmolecular weight 423.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16175
Actions Inhibitor
M. Wt 423.89
Formula C23H21N3O3.HCl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2002381-31-7
Synonyms KSR/Ras Inhibitor
SMILES CC1=C(C=CC(=C1)OC2=CC=CC=C2)NC3=NC=NC4=CC(=C(C=C43)OC)OC.Cl

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