ARV-771

Catalog No.: A13255
BET degrader
ARV-771 is a potent BET degrader based on PROTAC technology with Kds of 34, 4.7, 8.3, 7.6, 9.6, and 7.6 nM for BRD2(1), BRD2(2), BRD3(1), BRD3(2), BRD4(1), and BRD4(2), respectively.
Grouped product items
Product Name Price Stock Qty
ARV-771 1mg
$144.00
In stock
ARV-771 5mg
$432.00
In stock
ARV-771 10mg
$736.00
In stock
ARV-771 50mg
$2,208.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500

Important Notice: For research use only. We do not sell to patients.

Not your Region? View all Distributors

Adooq Products cited in reputable paper
Biological Activity
Discription ARV-771 is a potent BET degrader based on PROTAC technology with Kds of 34, 4.7, 8.3, 7.6, 9.6, and 7.6 nM for BRD2(1), BRD2(2), BRD3(1), BRD3(2), BRD4(1), and BRD4(2), respectively.
Targets
Target Value
Product Information
Catalog Num A13255
Formula C49H60ClN9O7S2
Molecular Weight 986.64
CAS Number 1949837-12-0
SMILES CC(C(C(C1=CC=C(Cl)C=C1)=N[C@@H](CC(NCCOCCCOCC(N[C@@H](C(C)(C)C)C(N(C[C@H](O)C2)[C@@H]2C(N[C@H](C3=CC=C(C(SC=N4)=C4C)C=C3)C)=O)=O)=O)=O)C5=NN=C(C)N65)=C6S7)=C7C
Synonyms ARV771, ARV 771
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 97 mg/mL (98.31 mM)
Water Insoluble
Ethanol 97 mg/mL (98.31 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 10.14 mL 50.68 mL 101.35 mL
0.5 mM 2.03 mL 10.14 mL 20.27 mL
1 mM 1.01 mL 5.07 mL 10.14 mL
5 mM 0.2 mL 1.01 mL 2.03 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2

  • Calculator Reset
Keywords: buy ARV-771 | ARV-771 Supplier | purchase ARV-771 | ARV-771 cost | ARV-771 manufacturer | order ARV-771 | ARV-771 distributor | buy 1949837-12-0 | 1949837-12-0 Supplier | purchase 1949837-12-0 | 1949837-12-0 cost | 1949837-12-0 manufacturer | order 1949837-12-0 | 1949837-12-0 distributor