Asenapine

Catalog No.: A18010

adrenergic receptor inhibitor

Asenapine

Asenapine Chemical Structure

CAS NO. 65576-45-6

Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM.

Availability: In stock

Package Price Qty
10 mg
$130.00
25 mg
$259.00
50 mg
$446.00
100 mg
$763.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 34.99 mL 174.97 mL 349.93 mL
0.5 mM 7 mL 34.99 mL 69.99 mL
1 mM 3.5 mL 17.5 mL 34.99 mL
5 mM 0.7 mL 3.5 mL 7 mL

*The above data is based on the productmolecular weight 285.77. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18010
Actions Inhibitor
CAS No. 65576-45-6
Formula C17H16ClNO
M. Wt 285.77
Purity >98%
Synonyms Org 5222, Org-5222, Org5222
SMILES ClC1=CC=C2OC3=CC=CC=C3[[email protected]@](C4)([H])[[email protected]](CN4C)([H])C2=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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