Atipamezole HCl

Catalog No.: A13902

α2 adrenergic receptor antagonist

Atipamezole HCl

Atipamezole HCl Chemical Structure

CAS NO. 104075-48-1

Atipamezole HCl is a selective α2-adrenergic receptor antagonist (Ki values are 1.1, 1.0, 0.89, 1300 and 6500 nM for α2A, α2B, α2C, α1A and α1B receptors respectively). Has been shown to be a brain penetrant.

Availability: In stock

Package Price Qty
10 mg
$90.00
25 mg
$200.00
50 mg
$300.00
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Biological Activity

Atipamezole HCl is a selective α2-adrenergic receptor antagonist (Ki values are 1.1, 1.0, 0.89, 1300 and 6500 nM for α2A, α2B, α2C, α1A and α1B receptors respectively). Has been shown to be a brain penetrant.
Targets
α2 adrenergic receptor
In vitro DMSO 12 mg/mL (48.24 mM)
Water 21 mg/mL (84.42 mM)
Ethanol 48 mg/mL (192.96 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 40.19 mL 200.96 mL 401.93 mL
0.5 mM 8.04 mL 40.19 mL 80.39 mL
1 mM 4.02 mL 20.1 mL 40.19 mL
5 mM 0.8 mL 4.02 mL 8.04 mL

*The above data is based on the productmolecular weight 248.8. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13902
Actions Antagonist
CAS No. 104075-48-1
Formula C14H16N2.HCl
M. Wt 248.8
Purity >98%
Synonyms Antisedan
SMILES CCC1(CC2=CC=CC=C2C1)C3=CN=CN3.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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