Avasimibe (CI-1011)

Catalog No.: A10102

CYP17 inhibitor

Avasimibe (CI-1011)

Avasimibe (CI-1011) Chemical Structure

CAS NO. 166518-60-1

Avasimibe (CI-1011) is an orally bioavailable Acyl-CoA:Cholesterol O-Acyltransferase (ACAT) inhibitor.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $50.00

Special Price $40.00

50 mg

Regular Price: $180.00

Special Price $144.00

100 mg

Regular Price: $320.00

Special Price $256.00

200 mg

Regular Price: $520.00

Special Price $416.00

10mM * 1mL in DMSO
$84.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

Avasimibe (CI-1011) is an orally bioavailable Acyl-CoA:Cholesterol O-Acyltransferase (ACAT) inhibitor.
Targets
CYP2C9 ACAT CYP1A2 CYP2C19
2.9 μM3.3 μM13.9 μM26.5 μM
In vitro (25°C) DMSO 100 mg/mL (199.31 mM
Water <1 mg/mL (<1 mM)
Ethanol 8 mg/mL (15.94 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.93 mL 99.66 mL 199.32 mL
0.5 mM 3.99 mL 19.93 mL 39.86 mL
1 mM 1.99 mL 9.97 mL 19.93 mL
5 mM 0.4 mL 1.99 mL 3.99 mL

*The above data is based on the productmolecular weight 501.7 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A10102
Actions Inhibitor
M. Wt 501.7
Formula C29H43NO4S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 166518-60-1
Synonyms CI-1011, CI1011, PD 148515
SMILES CC(C)C1=C(C(=CC=C1)C(C)C)OS(=O)(=O)NC(=O)CC2=C(C=C(C=C2C(C)C)C(C)C)C(C)C

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