Catalog No.: A20204

PAR2 antagonist


AZ3451 Chemical Structure

CAS NO. 2100284-59-9

AZ3451 is a potent protease-activated receptor-2 (PAR2) antagonist with IC50 of 23 nM.

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Biological Activity

AZ3451 is a potent protease-activated receptor-2 (PAR2) antagonist with IC50 of 23 nM.
In vitro DMSO 97 mg/mL (169.74 mM)
Water Insoluble
Ethanol 97 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.5 mL 87.5 mL 174.99 mL
0.5 mM 3.5 mL 17.5 mL 35 mL
1 mM 1.75 mL 8.75 mL 17.5 mL
5 mM 0.35 mL 1.75 mL 3.5 mL

*The above data is based on the productmolecular weight 571.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20204
Actions Antagonist
CAS No. 2100284-59-9
Formula C30H27BrN4O3
M. Wt 571.46
Purity >98%
Synonyms AZ 3451, AZ-3451
SMILES O=C(C1=CC=C2C(N=C(C3=C(Br)C=C(OCO4)C4=C3)N2[[email protected]](C5CCCCC5)C)=C1)NC6=CC=C(C#N)C=C6

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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