AZ505

Catalog No.: A13061

SMYD2 inhibitor

AZ505

AZ505 Chemical Structure

CAS NO. 1035227-43-0

AZ505 is a potent and highly selective inhibitor of the oncogenic protein SMYD2(IC50=0.12 μM) with potential anticancer activity, >600 fold than SMYD3(IC50>83.3 μM); DOT1L(IC50>83.3 μM);EZH2(IC50>83.3 μM).

Availability: In stock

Package Price Qty
5 mg
$180.00
10 mg
$320.00
50 mg
$960.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AZ505 is a potent and highly selective inhibitor of the oncogenic protein SMYD2(IC50=0.12 μM) with potential anticancer activity, >600 fold than SMYD3(IC50>83.3 μM); DOT1L(IC50>83.3 μM);EZH2(IC50>83.3 μM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.31 mL 86.57 mL 173.15 mL
0.5 mM 3.46 mL 17.31 mL 34.63 mL
1 mM 1.73 mL 8.66 mL 17.31 mL
5 mM 0.35 mL 1.73 mL 3.46 mL

*The above data is based on the productmolecular weight 577.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A13061
Actions Inhibitor
M. Wt 577.54
Formula C29H38Cl2N4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1035227-43-0
Synonyms AZ 505, AZ-505
SMILES C1CCC(CC1)N(CCNCCC2=C3C(=C(C=C2)O)NC(=O)CO3)C(=O)CCNCCC4=CC(=C(C=C4)Cl)Cl

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