Biological Activity
Azasetron HCl is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy.
In vitro | DMSO | Insoluble | |
Water | 3 mg/mL (7.76 mM) | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 25.89 mL | 129.44 mL | 258.89 mL |
0.5 mM | 5.18 mL | 25.89 mL | 51.78 mL |
1 mM | 2.59 mL | 12.94 mL | 25.89 mL |
5 mM | 0.52 mL | 2.59 mL | 5.18 mL |
*The above data is based on the productmolecular weight 386.27. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A16417 |
---|---|
Actions | Antagonist |
CAS No. | 123040-16-4 |
Formula | C17H20ClN3O3.HCl |
M. Wt | 386.27 |
Solubility | DMSO |
Purity | >98% |
Synonyms | Y-25130 hydrochloride, Y25130 hydrochloride, Y 25130 hydrochloride |
SMILES | CN1C(=O)COC2=C1C=C(C=C2C(=O)NC3CN4CCC3CC4)Cl.Cl |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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