Batefenterol

Catalog No.: A21387

muscarinic receptor antagonist and β2-adrenoceptor agonist

Batefenterol

Batefenterol Chemical Structure

CAS NO. 743461-65-6

Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively.

Availability: In stock

Package Price Qty
5 mg
$151.00
10 mg
$260.00
50 mg
$773.00
100 mg
$1,546.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 13.51 mL 67.55 mL 135.09 mL
0.5 mM 2.7 mL 13.51 mL 27.02 mL
1 mM 1.35 mL 6.75 mL 13.51 mL
5 mM 0.27 mL 1.35 mL 2.7 mL

*The above data is based on the productmolecular weight 740.24. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21387
Actions Antagonist
M. Wt 740.24
Formula C40H42ClN5O7
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 743461-65-6
Synonyms GSK961081, GSK-961081, GSK 961081; TD-5959, TD5959, TD 5959
SMILES O=C(OC1CCN(CCC(NC2=CC(OC)=C(CNC[[email protected]](O)C3=CC=C(O)C4=C3C=CC(N4)=O)C=C2Cl)=O)CC1)NC5=CC=CC=C5C6=CC=CC=C6

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Batefenterol | Batefenterol Supplier | purchase | cost | manufacturer | order | distributor | buy 743461-65-6| 743461-65-6 Supplier | purchase 743461-65-6 | 743461-65-6 cost | 743461-65-6 manufacturer | order 743461-65-6 | 743461-65-6 distributor
Rewards