Batefenterol

Catalog No.: A21387

muscarinic receptor antagonist and β2-adrenoceptor agonist

Batefenterol

Batefenterol Chemical Structure

CAS NO. 743461-65-6

Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively.

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5 mg

Regular Price: $151.00

Special Price $120.80

10 mg

Regular Price: $260.00

Special Price $208.00

50 mg

Regular Price: $773.00

Special Price $618.40

100 mg

Regular Price: $1,546.00

Special Price $1,236.80

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Biological Activity

Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 13.51 mL 67.55 mL 135.09 mL
0.5 mM 2.7 mL 13.51 mL 27.02 mL
1 mM 1.35 mL 6.75 mL 13.51 mL
5 mM 0.27 mL 1.35 mL 2.7 mL

*The above data is based on the productmolecular weight 740.24. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21387
Actions Antagonist
CAS No. 743461-65-6
Formula C40H42ClN5O7
M. Wt 740.24
Purity >98%
Synonyms GSK961081, GSK-961081, GSK 961081; TD-5959, TD5959, TD 5959
SMILES O=C(OC1CCN(CCC(NC2=CC(OC)=C(CNC[[email protected]](O)C3=CC=C(O)C4=C3C=CC(N4)=O)C=C2Cl)=O)CC1)NC5=CC=CC=C5C6=CC=CC=C6
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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