BETd-246

Catalog No.: A18913

BRD inhibitor

BETd-246

BETd-246 Chemical Structure

CAS NO. 2140289-17-2

BETd-246 is a second-generation BET bromodomain (BRD) inhibitor, exhibiting superior selectivity, potency and antitumor activity.

Availability: In stock

Package Price Qty
1 mg
$180.00
5 mg
$600.00
10 mg
$900.00
50 mg
$2,700.00
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Biological Activity

BETd-246 is a second-generation BET bromodomain (BRD) inhibitor, exhibiting superior selectivity, potency and antitumor activity.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 10.57 mL 52.85 mL 105.7 mL
0.5 mM 2.11 mL 10.57 mL 21.14 mL
1 mM 1.06 mL 5.29 mL 10.57 mL
5 mM 0.21 mL 1.06 mL 2.11 mL

*The above data is based on the productmolecular weight 946.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18913
Actions Inhibitor
CAS No. 2140289-17-2
Formula C48H55N11O10
M. Wt 946.03
Solubility DMSO
Purity >98%
Synonyms BETd-246; BETd 246; BETd246
SMILES O=C(C1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1)NCCCOCCOCCOCCCNC7=CC=CC(C(N8C(CC9)C(NC9=O)=O)=O)=C7C8=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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