BETd-260

Catalog No.: A12563

BET degrader

BETd-260

BETd-260 Chemical Structure

CAS NO. 2093388-62-4

BETd-260 is a potent BET degrader based on PROTAC technology, with as low as 30 pM against BRD4 protein in RS4;11 leukemia cell line.

Availability: In stock

Package Price Qty
5 mg
$405.00
10 mg
$698.00
50 mg
$2,070.00
100 mg
$4,140.00
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Biological Activity

BETd-260 is a potent BET degrader based on PROTAC technology, with as low as 30 pM against BRD4 protein in RS4;11 leukemia cell line.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.52 mL 62.59 mL 125.17 mL
0.5 mM 2.5 mL 12.52 mL 25.03 mL
1 mM 1.25 mL 6.26 mL 12.52 mL
5 mM 0.25 mL 1.25 mL 2.5 mL

*The above data is based on the productmolecular weight 798.89. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12563
Actions Degrader
CAS No. 2093388-62-4
Formula C43H46N10O6
M. Wt 798.89
Purity >98%
Synonyms BETd260, BETd 260, ZBC 260, ZBC-260, ZBC260
SMILES CCN1N=C(C2CC2)C=C1NC3=NC(C(NCCCCCC4=CC=CC5=C4CN(C6C(NC(CC6)=O)=O)C5=O)=O)=NC7=C3C8=CC(OC)=C(C9=C(C)ON=C9C)C=C8N7
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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